99% Cetilistat CAS Lamba 282526-98-1
Suna: Cetilistat
Bayyanar: Ƙirjin da ba ya da fari.
Lambar CAS: 282526-98-1
Yawan yawa: 1.027 g/cm3
Tsarin dabara: C25H39NO3
Tafasawar Teku: 509.671 °C a 760 mmHg
Nauyin kwayoyin halitta: 401.58
Wurin Wahala: 158.925 °C
Ma'anar kalmomi: 2-(Hexadecyloxy)-6-methyl-4H-3,1-benzoxazin-4-one
The Cetilistat wani sinadari ne na halitta wanda ke ɗauke da dabarar C25H39NO3. Sunan IUPAC na wannan sinadari shine 2-hexadecoxy-6-methyl-3,1-benzoxazin-4-one. Tare da lambar rajista ta CAS 282526-98-1, ana kuma kiransa da 4H-3,1-benzoxazin-4-one, 2-(hexadecyloxy)-6-methyl-. Lambar rarrabuwar samfurin ita ce Maganin kiba. Bugu da ƙari, magani ne da aka tsara don magance kiba. Yana aiki kamar yadda yake a da, orlistat, magani na da, ta hanyar hana pancreas lipase, wani enzyme da ke rushe triglycerides a cikin hanji. Ba tare da wannan enzyme ba, ana hana triglycerides daga abinci su zama acid mai kitse mai narkewa kuma ana fitar da su ba tare da narkewa ba.
Cetilistat magani ne da aka ƙera don magance kiba. Yana aiki kamar yadda aka ƙera da daɗaɗɗen magani orlistat (Xenical) ta hanyar hana pancreas lipase, wani enzyme wanda ke rushe triglycerides a cikin hanji. Ba tare da wannan enzyme ba, ana hana triglycerides daga abinci su zama fatty acids masu narkewa kuma ana fitar da su ba tare da narkewa ba.
A cikin gwaje-gwajen da aka yi wa mutane, an nuna cewa Cetilistat yana haifar da irin wannan asarar nauyi kamar orlistat, amma kuma yana haifar da irin waɗannan illoli kamar mai, bayan gida mai laushi, rashin kwanciyar hankali a cikin najasa, yawan motsa hanji, da kuma kumburin ciki. Akwai yiwuwar irin waɗannan matakan za a yi amfani da su wajen hana shan bitamin masu narkewar mai da sauran abubuwan gina jiki masu narkewar mai, wanda ke buƙatar a yi amfani da ƙarin bitamin don guje wa rashi.
| Tsarin Aiki: Tsarin Kasuwanci | |
| KAYAN BINCIKE | MAS'ALA |
| Bayyanar | Foda fari zuwa launin ruwan kasa |
| Ganowa | Ya dace |
| ruwa | ≤0.5% |
| Sauran sinadaran da ke narkewa | Acetone ≤5000ppm |
| Acetonitrile≤410ppm | |
| Karfe masu nauyi | ≤20ppm |
| HPLC | ≥99.0% |
| Rashin tsarki guda ɗaya | ≤0.2% |
| Ragowar Wutar Lantarki | ≤0.2% |
| Kammalawa | Ya yi daidai da Ma'aunin Kasuwanci |









