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Fakitale ya GMP imapereka 99% min Triptorelin acetate cas yapamwamba kwambiri 140194-24-7

Kufotokozera Kwachidule:


Tsatanetsatane wa Zamalonda

Ma tag a Zamalonda

Mafotokozedwe Akatundu

Fakitale ya GMP imapereka 99% min Triptorelin acetate cas yapamwamba kwambiri 140194-24-7

Tsatanetsatane wa malonda:
Dzina la Mankhwala: Triptorelin acetate

Nambala ya CAS: 140194-24-7

Mafotokozedwe Ena Ofanana

Mau Oyamba:
Triptorelin ndi gonadotropin releasing hormone (GnRH) agonist yomwe ndi yoletsa kwambiri kupanga kwa estrogen (mwa akazi) ndipo imagwiritsidwa ntchito pochiza khansa ya prostate yoopsa.
Ndi D-tryptophan m'malo mwa residue 6.

Ndi mankhwala omwe amachititsa kuti pituitary iyambe kugwira ntchito, motero amachepetsa kutulutsa kwa luteinizing hormone (LH) ndi follicle stimulating hormone (FSH).
Triptorelin ndi decapeptide (pGlu-His-Trp-Ser-Tyr-D-Trp-Leu-Arg-Pro-Gly-NH2) ndi gonadotropin-releasing hormone agonist (GnRH agonist) yomwe imagwiritsidwa ntchito ngati acetate kapena pamoate salts.

Mapulogalamu:
Monga ma agonist ena a GnRH, triptorelin ingagwiritsidwe ntchito pochiza khansa yokhudzana ndi mahomoni monga khansa ya prostate kapena khansa ya m'mawere, kutha msinkhu msanga, matenda odalira estrogen.
(monga endometriosis kapena uterine fibroids), komanso mu chithandizo chothandizira kubereka.

Kulongedza:
1g/botolo, kapena malinga ndi zomwe mukufuna.
Iyenera kusungidwa pamalo ouma, ozizira komanso opumira mpweya, pewani kuzizira ndi chinyezi, isungeni kutali ndi ma oxides

Kufotokozera

CHINTHU
INDEX
Makhalidwe
ufa woyera wa kristalo
Kuyesa (HPLC)
≥99%
Kusayera Kokha (HPLC)
≤1.0%
Kapangidwe ka Amino Acid
± 10% ya mfundo zamaganizo
Kuchuluka kwa Peptide (N%)
≥80%
Kuchuluka kwa Madzi (Karl Fischer)
≤6.0%
Zomwe Zili mu Acetate (HPIC)
≤15.0%
MS(ESI)
Kugwirizana
Kuchuluka kwa Misa
95.0~105.0%
Kuzungulira Kwapadera (20/D)
-65.0~-75.0°(c=0.5 1%HAc)
* Kuphatikiza apo: Kampaniyo ikhoza kufufuza ndikupanga zinthu zatsopano malinga ndi zosowa zapadera za makasitomala athu.

 


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