mureza

chigadzirwa

Fekitori yeGMP inopa mhando yepamusoro ye99% min Triptorelin acetate cas 140194-24-7

Tsananguro pfupi:


Ruzivo rweChigadzirwa

Matagi eChigadzirwa

Tsananguro yeChigadzirwa

Fekitori yeGMP inopa mhando yepamusoro ye99% min Triptorelin acetate cas 140194-24-7

Ruzivo rwechigadzirwa:
Zita reKemikari: Triptorelin acetate

Nhamba yeCAS: 140194-24-7

Dzimwe Tsananguro Dzakabatana

Sumo:
Triptorelin ihormone inoburitsa gonadotropin (GnRH) agonist iyo inodzivirira kugadzirwa kweestrogen (muvakadzi) uye inoshandiswa kurapa kenza yeprostate yakakwira.
Inotsiva D-tryptophan pane residue 6.

Mushonga unokonzera kukurudzira kwepituitary, nokudaro uchideredza kuburitswa kwehomoni yeluteinizing (LH) uye homoni inokurudzira follicle (FSH).
Triptorelin idecapeptide (pGlu-His-Trp-Ser-Tyr-D-Trp-Leu-Arg-Pro-Gly-NH2) uye gonadotropin-releasing hormone agonist (GnRH agonist) inoshandiswa se acetate kana pamoate salts.

Mashandisirwo:
Kufanana nedzimwe agonist dzeGnRH, triptorelin inogona kushandiswa mukurapa kenza dzinopindura mahormone dzakadai sekenza yeprostate kana kenza yemazamu, kuyaruka kwepakutanga, uye mamiriro ezvinhu anoenderana neestrogen.
(senge endometriosis kana uterine fibroids), uye mukubatsira kubereka.

Kurongedza:
1g/bhodhoro, kana zvichienderana nezvaunoda.
Inofanira kuchengetwa munzvimbo yakaoma, inotonhorera uye ine mhepo, kudzivirira kusviba uye hunyoro, ichengete kure nema oxides

Tsanangudzo

CHINHU
INDEX
Hunhu
upfu chena hwekristaro
Kuyedza (HPLC)
≥99%
Kusachena Kumwechete (HPLC)
≤1.0%
Kuumbwa kweAmino Acid
±10% yedzidziso
Zviri Mukati mePeptide (N%)
≥80%
Zviri Mumvura (Karl Fischer)
≤6.0%
Zviri MuAcetate (HPIC)
≤15.0%
MS(ESI)
Kugara kuripo
Kuenzana Kwehuwandu
95.0~105.0%
Kutenderera Kwakananga (20/D)
-65.0~-75.0°(c=0.5 1%HAc)
* Pamusoro pezvo: Kambani inogona kutsvagisa nekugadzira zvigadzirwa zvitsva zvichienderana nekudiwa kwakakosha kwevatengi vedu.

 


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