Warshadda GMP waxay bixisaa tayo sare leh 99% daqiiqo Triptorelin acetate cas 140194-24-7
Warshadda GMP waxay bixisaa tayo sare leh 99% daqiiqo Triptorelin acetate cas 140194-24-7
Faahfaahinta alaabta:
Magaca Kiimikada: Triptorelin acetate
Lambarka CAS: 140194-24-7
Hordhacyo:
Triptorelin waa agonist hormoon sii daaya gonadotropin (GnRH) kaas oo ah mid si xooggan u xakameeya isku-darka estrogen (haweenka) waxaana loo isticmaalaa in lagu daaweeyo kansarka qanjirka 'prostate' ee horumarsan.
Waa beddel D-tryptophan ah marka la barbar dhigo residue 6.
Waa daawo keenta kicinta qanjirka 'pituitary', taasoo hoos u dhigaysa soo saarista hoormoonka luteinizing (LH) iyo hoormoonka kicinta follicle (FSH).
Triptorelin waa decapeptide (pGlu-His-Trp-Ser-Tyr-D-Trp-Leu-Arg-Pro-Gly-NH2) iyo agonist hoormoonka sii daaya gonadotropin (agonist GnRH) oo loo isticmaalo cusbada acetate ama pamoate.
Codsiyada:
Sida daawooyinka kale ee GnRH agonists, triptorelin waxaa loo isticmaali karaa daaweynta kansarka ka jawaaba hoormoonka sida kansarka qanjirka 'prostate' ama kansarka naasaha, qaangaarnimada hore, xaaladaha ku tiirsan estrogen-ka.
(sida endometriosis ama fibroids ilmo-galeenka), iyo taranka caawinta.
Baakad:
1g/dhalo, ama sida aad u baahan tahay.
Waa in lagu kaydiyaa meel qalalan, qabow oo hawo leh, iska ilaali qoyaanka iyo qoyaanka, ka fogee oksaydhyada.
| SHAYGA | TUSMADA |
| Astaamaha | budada kristalinta cad |
| Baaritaan (HPLC) | ≥99% |
| Nadaafad Keli ah (HPLC) | ≤1.0% |
| Halabuurka Asiidhka Amino | ±10% ee aragtiyeedka |
| Waxyaabaha ku jira Peptide (N%) | ≥80% |
| Biyaha ku jira (Karl Fischer) | ≤6.0% |
| Maaddada Acetate (HPIC) | ≤15.0% |
| MS(ESI) | Joogto ah |
| Isu-dheellitirka Cufnaanta | 95.0~105.0% |
| Wareeg Gaar ah (20/D) | -65.0~-75.0°(c=0.5 1%HAc) |
| * Intaa waxaa dheer: Shirkaddu waxay baari kartaa oo horumarin kartaa alaabada cusub iyadoo loo eegayo baahida gaarka ah ee macaamiisheenna. | |









