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Warshadda GMP waxay bixisaa tayo sare leh 99% daqiiqo Triptorelin acetate cas 140194-24-7

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Calaamadaha Alaabta

Sharaxaadda Badeecada

Warshadda GMP waxay bixisaa tayo sare leh 99% daqiiqo Triptorelin acetate cas 140194-24-7

Faahfaahinta alaabta:
Magaca Kiimikada: Triptorelin acetate

Lambarka CAS: 140194-24-7

Sharaxaadaha Kale ee La Xiriira

Hordhacyo:
Triptorelin waa agonist hormoon sii daaya gonadotropin (GnRH) kaas oo ah mid si xooggan u xakameeya isku-darka estrogen (haweenka) waxaana loo isticmaalaa in lagu daaweeyo kansarka qanjirka 'prostate' ee horumarsan.
Waa beddel D-tryptophan ah marka la barbar dhigo residue 6.

Waa daawo keenta kicinta qanjirka 'pituitary', taasoo hoos u dhigaysa soo saarista hoormoonka luteinizing (LH) iyo hoormoonka kicinta follicle (FSH).
Triptorelin waa decapeptide (pGlu-His-Trp-Ser-Tyr-D-Trp-Leu-Arg-Pro-Gly-NH2) iyo agonist hoormoonka sii daaya gonadotropin (agonist GnRH) oo loo isticmaalo cusbada acetate ama pamoate.

Codsiyada:
Sida daawooyinka kale ee GnRH agonists, triptorelin waxaa loo isticmaali karaa daaweynta kansarka ka jawaaba hoormoonka sida kansarka qanjirka 'prostate' ama kansarka naasaha, qaangaarnimada hore, xaaladaha ku tiirsan estrogen-ka.
(sida endometriosis ama fibroids ilmo-galeenka), iyo taranka caawinta.

Baakad:
1g/dhalo, ama sida aad u baahan tahay.
Waa in lagu kaydiyaa meel qalalan, qabow oo hawo leh, iska ilaali qoyaanka iyo qoyaanka, ka fogee oksaydhyada.

Faahfaahinta

SHAYGA
TUSMADA
Astaamaha
budada kristalinta cad
Baaritaan (HPLC)
≥99%
Nadaafad Keli ah (HPLC)
≤1.0%
Halabuurka Asiidhka Amino
±10% ee aragtiyeedka
Waxyaabaha ku jira Peptide (N%)
≥80%
Biyaha ku jira (Karl Fischer)
≤6.0%
Maaddada Acetate (HPIC)
≤15.0%
MS(ESI)
Joogto ah
Isu-dheellitirka Cufnaanta
95.0~105.0%
Wareeg Gaar ah (20/D)
-65.0~-75.0°(c=0.5 1%HAc)
* Intaa waxaa dheer: Shirkaddu waxay baari kartaa oo horumarin kartaa alaabada cusub iyadoo loo eegayo baahida gaarka ah ee macaamiisheenna.

 


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