ibhena

umkhiqizo

Intengo enhle Izithako zemithi eziphakathi 99% Nicergoline CAS 27848-84-6

Incazelo emfushane:


Imininingwane Yomkhiqizo

Amathegi Omkhiqizo

Incazelo Yomkhiqizo

Intengo enhle Izithako zemithi eziphakathi 99% Nicergoline CAS 27848-84-6

Imininingwane yomkhiqizo:
Igama Lekhemikhali: I-Nicergoline

Ifomula Yamamolekyuli:C24H26BrN3O3

Inombolo ye-CAS: 27848-84-6

Ibanga: CP/EP/USP

Ezinye Izincazelo Ezihlobene

Isingeniso:
I-Nicergoline, njengoSermion, uJoseph Hermione, i-nicergoline, uKell; uwine ikhemikhali yokuqala ye-ninni cabergoline ebizwa ngokuthi i-alpha 10 methoxy two methyl -1,6- cabergoline -8 beta 5''-nicotinate. Ifomula yama-molecule esekelwe ku-Bromine methanol: c24h26brn3o3 isisindo sama-molecule singama-484.39. noma izinkomba ezibukhali ukuphazamiseka kwe-cerebrovascular okungapheli noma ukungasebenzi kahle kwe-metabolic yobuchopho. Ukuhamba, ukungasebenzi kahle kobuchopho okungapheli okubangelwa yizithiyo zolimi, isiyezi, i-tinnitus, umbono ofiphele, umuzwa, ikhanda elibuhlungu, ukungakwazi ukulala, ukulahlekelwa yinkumbulo, ukunganaki, ukucindezeleka, ukukhathazeka, injabulo kanye ne-dementia. Amaphilisi e-Nicergoline angathuthukisa umsebenzi wezidakamizwa zokwehlisa umfutho wegazi. Ngenxa yokuthi i-nicergoline iguqulwa yi-CytochromeP4502D6, ayikukhiphi ukusebenzisana nezidakamizwa ngendlela efanayo.

Imisebenzi:
1. I-Nicergoline iyi-dervitus ye-ergot esetshenziselwa ukwelapha i-senile dementia kanye nezinye izifo ezibangelwa yimithambo yegazi.

2. Kutholakale ukuthi kwandisa ukuguquguquka kwengqondo nokuthuthukisa ukucaca nokuqonda.

3. Kunciphisa ukumelana kwemithambo yegazi futhi kwandisa ukugeleza kwegazi ebuchosheni, kuthuthukisa ukusetshenziswa komoya-mpilo kanye ne-glucose ngamaseli obuchopho.

4. Inezakhiwo ezifanayo zokuvuselela amasosha omzimba kwezinye izindawo zomzimba, ikakhulukazi amaphaphu.

5. Isetshenziselwa izifo zemithambo yegazi ezifana ne-cerebral thrombosis kanye ne-atherosclerosis, ukuvaleka kwemithambo yegazi emalungeni, isifo sikaRaynaud, i-vascular migraines, kanye ne-retinopathy.

6. I-Nicergoline ibhaliswe emazweni angaphezu kwamashumi amahlanu futhi isetshenziswe iminyaka engaphezu kwamashumi amathathu ekwelapheni ukuphazamiseka kwengqondo, ukuzwela, kanye nokuziphatha kwabantu asebekhulile.

Ukupakisha:
isikhwama sepulasitiki ngaphakathi kanye nesikhwama se-aluminium ngaphandle
Indawo yokugcina: Emthunzini omnyama nesimo. Kanye nokushisa okuphansi (+2--+8ºC)

Imininingwane

ITEM
I-INDEX
Izici
Ikristalu elimhlophe noma i-powder
Indawo yokuncibilika
133ºC ~ 136ºC
Ukujikeleza okubonakalayo okuqondile
Ukuhambisana
Ukucaca nombala wesisombululo
Sula
Izinto ezihlobene
Ukungcola okuphelele ≤1.5%
I-Nor-nocergoline (B) ≤0.50%
I-Chioronicergoline (A) ≤0.5%
I-MeLUOL (C) ≤0.30%
Ukungcola okungaziwa: ≤0.30%
Amanzi
≤0.5%
Insimbi enamandla
≤20ppm
Izinsalela ezivuthayo
≤0.05%
Ukuhlolwa
98.5% ~ 102%
Izithasiselo ezisele
I-Acetone
≤1000ppm
I-ether ye-Diethyl
≤2000ppm
I-Ethanol
≤1000ppm
I-Methanol
≤1000ppm
I-Toluene
≤500ppm
I-Dichloromethan
≤100ppm
I-Triethylamine
≤500ppm
Isiphetho
Vumelana ne-EP 5.0
* Ngaphezu kwalokho: Inkampani ingacwaninga futhi ithuthukise imikhiqizo emisha ngokwesidingo esikhethekile samakhasimende ethu.

 


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