Intengo enhle Izithako zemithi eziphakathi 99% Nicergoline CAS 27848-84-6
Intengo enhle Izithako zemithi eziphakathi 99% Nicergoline CAS 27848-84-6
Imininingwane yomkhiqizo:
Igama Lekhemikhali: I-Nicergoline
Ifomula Yamamolekyuli:C24H26BrN3O3
Inombolo ye-CAS: 27848-84-6
Ibanga: CP/EP/USP
Isingeniso:
I-Nicergoline, njengoSermion, uJoseph Hermione, i-nicergoline, uKell; uwine ikhemikhali yokuqala ye-ninni cabergoline ebizwa ngokuthi i-alpha 10 methoxy two methyl -1,6- cabergoline -8 beta 5''-nicotinate. Ifomula yama-molecule esekelwe ku-Bromine methanol: c24h26brn3o3 isisindo sama-molecule singama-484.39. noma izinkomba ezibukhali ukuphazamiseka kwe-cerebrovascular okungapheli noma ukungasebenzi kahle kwe-metabolic yobuchopho. Ukuhamba, ukungasebenzi kahle kobuchopho okungapheli okubangelwa yizithiyo zolimi, isiyezi, i-tinnitus, umbono ofiphele, umuzwa, ikhanda elibuhlungu, ukungakwazi ukulala, ukulahlekelwa yinkumbulo, ukunganaki, ukucindezeleka, ukukhathazeka, injabulo kanye ne-dementia. Amaphilisi e-Nicergoline angathuthukisa umsebenzi wezidakamizwa zokwehlisa umfutho wegazi. Ngenxa yokuthi i-nicergoline iguqulwa yi-CytochromeP4502D6, ayikukhiphi ukusebenzisana nezidakamizwa ngendlela efanayo.
Imisebenzi:
1. I-Nicergoline iyi-dervitus ye-ergot esetshenziselwa ukwelapha i-senile dementia kanye nezinye izifo ezibangelwa yimithambo yegazi.
2. Kutholakale ukuthi kwandisa ukuguquguquka kwengqondo nokuthuthukisa ukucaca nokuqonda.
3. Kunciphisa ukumelana kwemithambo yegazi futhi kwandisa ukugeleza kwegazi ebuchosheni, kuthuthukisa ukusetshenziswa komoya-mpilo kanye ne-glucose ngamaseli obuchopho.
4. Inezakhiwo ezifanayo zokuvuselela amasosha omzimba kwezinye izindawo zomzimba, ikakhulukazi amaphaphu.
5. Isetshenziselwa izifo zemithambo yegazi ezifana ne-cerebral thrombosis kanye ne-atherosclerosis, ukuvaleka kwemithambo yegazi emalungeni, isifo sikaRaynaud, i-vascular migraines, kanye ne-retinopathy.
6. I-Nicergoline ibhaliswe emazweni angaphezu kwamashumi amahlanu futhi isetshenziswe iminyaka engaphezu kwamashumi amathathu ekwelapheni ukuphazamiseka kwengqondo, ukuzwela, kanye nokuziphatha kwabantu asebekhulile.
Ukupakisha:
isikhwama sepulasitiki ngaphakathi kanye nesikhwama se-aluminium ngaphandle
Indawo yokugcina: Emthunzini omnyama nesimo. Kanye nokushisa okuphansi (+2--+8ºC)
| ITEM | I-INDEX |
| Izici | Ikristalu elimhlophe noma i-powder |
| Indawo yokuncibilika | 133ºC ~ 136ºC |
| Ukujikeleza okubonakalayo okuqondile | Ukuhambisana |
| Ukucaca nombala wesisombululo | Sula |
| Izinto ezihlobene | Ukungcola okuphelele ≤1.5% I-Nor-nocergoline (B) ≤0.50% I-Chioronicergoline (A) ≤0.5% I-MeLUOL (C) ≤0.30% Ukungcola okungaziwa: ≤0.30% |
| Amanzi | ≤0.5% |
| Insimbi enamandla | ≤20ppm |
| Izinsalela ezivuthayo | ≤0.05% |
| Ukuhlolwa | 98.5% ~ 102% |
| Izithasiselo ezisele | |
| I-Acetone | ≤1000ppm |
| I-ether ye-Diethyl | ≤2000ppm |
| I-Ethanol | ≤1000ppm |
| I-Methanol | ≤1000ppm |
| I-Toluene | ≤500ppm |
| I-Dichloromethan | ≤100ppm |
| I-Triethylamine | ≤500ppm |
| Isiphetho | Vumelana ne-EP 5.0 |
| * Ngaphezu kwalokho: Inkampani ingacwaninga futhi ithuthukise imikhiqizo emisha ngokwesidingo esikhethekile samakhasimende ethu. | |









