Feme ea GMP e fana ka boleng bo holimo ba 99% min Triptorelin acetate cas 140194-24-7
Feme ea GMP e fana ka boleng bo holimo ba 99% min Triptorelin acetate cas 140194-24-7
Lintlha tsa sehlahisoa:
Lebitso la Lik'hemik'hale: Triptorelin acetate
Nomoro ea CAS: 140194-24-7
Likenyelletso:
Triptorelin ke agonist ea gonadotropin releasing hormone (GnRH) e leng thibelo e matla ea tlhahiso ea estrogen (ho basali) 'me e sebelisetsoa ho phekola mofetše o tsoetseng pele oa tšoelesa ea senya.
Ke sebaka sa D-tryptophan ho masala a 6.
Ke moriana o bakang tlhohlelletso ea pituitary, ka hona o fokotsa ho ntšoa ha hormone ea luteinizing (LH) le hormone e susumetsang follicle (FSH).
Triptorelin ke decapeptide (pGlu-His-Trp-Ser-Tyr-D-Trp-Leu-Arg-Pro-Gly-NH2) le gonadotropin-releasing hormone agonist (GnRH agonist) e sebediswang e le acetate kapa pamoate salts.
Likopo:
Joalo ka li-agonist tse ling tsa GnRH, triptorelin e ka sebelisoa kalafong ea mofetše o arabelang lihormone joalo ka mofetše oa tšoelesa ea senya kapa mofetše oa matsoele, bohlankana ba pele ho nako, le maemo a itšetlehileng ka estrogen.
(joalo ka endometriosis kapa uterine fibroids), le ho thusoeng ho ikatisa.
Pakete:
1g/botlolo, kapa ho ya ka tlhoko ya hao.
E lokela ho bolokoa sebakeng se omileng, se pholileng le se nang le moea o mongata, qoba ho fifala le mongobo, e boloke hole le li-oxide.
| NTHO | INDEX |
| Litšobotsi | phofo e tšoeu ea kristale |
| Teko (HPLC) | ≥99% |
| Litšila tse le 'Ngoe (HPLC) | ≤1.0% |
| Sebopeho sa Amino Acid | ± 10% ea khopolo-taba |
| Dikahare tsa Peptide (N%) | ≥80% |
| Sekhahla sa Metsi (Karl Fischer) | ≤6.0% |
| Dikahare tsa Acetate (HPIC) | ≤15.0% |
| MS(ESI) | E tsitsitseng |
| Tekanyo ea Boima | 95.0~105.0% |
| Potoloho e Ikhethang (20/D) | -65.0~-75.0°(c=0.5 1%HAc) |
| * Ho phaella moo: Khamphani e ka etsa lipatlisiso le ho ntshetsa pele dihlahiswa tse ntjha ho ya ka tlhoko e ikgethang ya bareki ba rona. | |









