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Ụlọ ọrụ mmepụta ihe GMP na-enye ezigbo mma 99% nkeji Triptorelin acetate cas 140194-24-7

Nkọwa Dị Mkpirikpi:


Nkọwa Ngwaahịa

Akara Ngwaahịa

Nkọwa Ngwaahịa

Ụlọ ọrụ mmepụta ihe GMP na-enye ezigbo mma 99% nkeji Triptorelin acetate cas 140194-24-7

Nkọwa ngwaahịa:
Aha kemịkalụ: Triptorelin acetate

Nọmba CAS: 140194-24-7

Nkọwa Ndị Ọzọ Yiri Ya

Okwu Mmalite:
Triptorelin bụ ọgwụ na-eme ka hormone nke na-ewepụta gonadotropin (GnRH) dị ike nke na-egbochi mmepụta estrogen (n'ime ụmụ nwanyị) ma a na-ejikwa ya agwọ ọrịa kansa prostate dị elu.
Ọ bụ nnọchi D-tryptophan na residue 6.

Ọ bụ ọgwụ na-akpali pituitary, si otú a na-ebelata mmepụta nke hormone luteinizing (LH) na hormone na-akpali akpali (FSH).
Triptorelin bụ decapeptide (pGlu-His-Trp-Ser-Tyr-D-Trp-Leu-Arg-Pro-Gly-NH2) na gonadotropin-releasing hormone agonist (GnRH agonist) nke a na-eji dị ka acetate ma ọ bụ pamoate salts.

Ngwa:
Dịka ndị ọzọ na-agwọ ọrịa GnRH, enwere ike iji triptorelin gwọọ kansa ndị na-anabata homonu dịka kansa prostate ma ọ bụ kansa ara, afọ ime tupu oge eruo, na ọnọdụ dabere na estrogen.
(dịka endometriosis ma ọ bụ fibroids nke akpanwa), nakwa n'inyere aka n'ịmụpụta nwa.

Nkwakọba:
1g/karama, ma ọ bụ dịka ihe ị chọrọ.
A ga-echekwa ya n'ebe kpọrọ nkụ, dị jụụ ma dị jụụ, zere insolation na mmiri, debe ya n'ebe dị anya site na oxides.

Nkọwapụta

IHE
NTỤKWASỊ
Àgwà
ntụ ntụ kristal ọcha
Nnyocha (HPLC)
≥99%
Nchacha Otu (HPLC)
≤1.0%
Ngwakọta Amino Acid
±10% nke usoro echiche
Ọdịnaya Peptide (N%)
≥80%
Mmiri dị n'ime ya (Karl Fischer)
≤6.0%
Ọdịnaya Acetate (HPIC)
≤15.0%
MS(ESI)
Na-agbanwe agbanwe
Nhazi Oke
95.0~105.0%
Mgbanwe Pụrụ Iche (20/D)
-65.0~-75.0°(c=0.5 1%HAc)
* Na mgbakwunye: ụlọ ọrụ ahụ nwere ike inyocha ma mepụta ngwaahịa ọhụrụ dịka mkpa pụrụ iche nke ndị ahịa anyị siri dị.

 


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