Ụlọ ọrụ mmepụta ihe GMP na-enye ezigbo mma 99% nkeji Triptorelin acetate cas 140194-24-7
Ụlọ ọrụ mmepụta ihe GMP na-enye ezigbo mma 99% nkeji Triptorelin acetate cas 140194-24-7
Nkọwa ngwaahịa:
Aha kemịkalụ: Triptorelin acetate
Nọmba CAS: 140194-24-7
Okwu Mmalite:
Triptorelin bụ ọgwụ na-eme ka hormone nke na-ewepụta gonadotropin (GnRH) dị ike nke na-egbochi mmepụta estrogen (n'ime ụmụ nwanyị) ma a na-ejikwa ya agwọ ọrịa kansa prostate dị elu.
Ọ bụ nnọchi D-tryptophan na residue 6.
Ọ bụ ọgwụ na-akpali pituitary, si otú a na-ebelata mmepụta nke hormone luteinizing (LH) na hormone na-akpali akpali (FSH).
Triptorelin bụ decapeptide (pGlu-His-Trp-Ser-Tyr-D-Trp-Leu-Arg-Pro-Gly-NH2) na gonadotropin-releasing hormone agonist (GnRH agonist) nke a na-eji dị ka acetate ma ọ bụ pamoate salts.
Ngwa:
Dịka ndị ọzọ na-agwọ ọrịa GnRH, enwere ike iji triptorelin gwọọ kansa ndị na-anabata homonu dịka kansa prostate ma ọ bụ kansa ara, afọ ime tupu oge eruo, na ọnọdụ dabere na estrogen.
(dịka endometriosis ma ọ bụ fibroids nke akpanwa), nakwa n'inyere aka n'ịmụpụta nwa.
Nkwakọba:
1g/karama, ma ọ bụ dịka ihe ị chọrọ.
A ga-echekwa ya n'ebe kpọrọ nkụ, dị jụụ ma dị jụụ, zere insolation na mmiri, debe ya n'ebe dị anya site na oxides.
| IHE | NTỤKWASỊ |
| Àgwà | ntụ ntụ kristal ọcha |
| Nnyocha (HPLC) | ≥99% |
| Nchacha Otu (HPLC) | ≤1.0% |
| Ngwakọta Amino Acid | ±10% nke usoro echiche |
| Ọdịnaya Peptide (N%) | ≥80% |
| Mmiri dị n'ime ya (Karl Fischer) | ≤6.0% |
| Ọdịnaya Acetate (HPIC) | ≤15.0% |
| MS(ESI) | Na-agbanwe agbanwe |
| Nhazi Oke | 95.0~105.0% |
| Mgbanwe Pụrụ Iche (20/D) | -65.0~-75.0°(c=0.5 1%HAc) |
| * Na mgbakwunye: ụlọ ọrụ ahụ nwere ike inyocha ma mepụta ngwaahịa ọhụrụ dịka mkpa pụrụ iche nke ndị ahịa anyị siri dị. | |









